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Chun Wu
Chun Wu
Guangzhou Institutes of Biomedicine and Health
Chemistry
Prostate cancer
Cancer research
Bromodomain
Biochemistry
5
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71
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Y06014 is a selective BET inhibitor for the treatment of prostate cancer.
2021
Acta Pharmacologica Sinica
Tian-Bang Wu
Qiuping Xiang
Chao Wang
Chun Wu
Cheng Zhang
Zhang Maofeng
Liu Zhaoxuan
Yan Zhang
Lin-jiu Xiao
Yong Xu
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Citations (2)
Structure-Based Discovery and Optimization of Benzo[ d]isoxazole Derivatives as Potent and Selective BET Inhibitors for Potential Treatment of Castration-Resistant Prostate Cancer (CRPC)
2018
Journal of Medicinal Chemistry
Maofeng Zhang
Yan Zhang
Ming Song
Xiaoqian Xue
Junjian Wang
Chao Wang
Cheng Zhang
Chenchang Li
Qiuping Xiang
Lingjiao Zou
Xishan Wu
Chun Wu
Baijun Dong
Wei Xue
Yulai Zhou
Hongwu Chen
Donghai Wu
Ke Ding
Yong Xu
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Citations (22)
Discovery and optimization of 1-(1H-indol-1-yl)ethanone derivatives as CBP/EP300 bromodomain inhibitors for the treatment of castration-resistant prostate cancer.
2018
European Journal of Medicinal Chemistry
Qiuping Xiang
Chao Wang
Yan Zhang
Xiaoqian Xue
Ming Song
Cheng Zhang
Chenchang Li
Chun Wu
Kuai Li
Xiaoyan Hui
Yulai Zhou
Jeff B. Smaill
Adam V. Patterson
Donghai Wu
Ke Ding
Yong Xu
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Citations (31)
Y08060: A Selective BET Inhibitor for Treatment of Prostate Cancer
2018
ACS Medicinal Chemistry Letters
Qiuping Xiang
Yan Zhang
Jiaguo Li
Xiaoqian Xue
Chao Wang
Ming Song
Cheng Zhang
Rui Wang
Chenchang Li
Chun Wu
Yulai Zhou
Xiaohong Yang
Guohui Li
Ke Ding
Yong Xu
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Citations (8)
Discovery and structural optimization of 4-(4-(benzyloxy)phenyl)-3,4-dihydropyrimidin-2(1H)-ones as RORc inverse agonists
2016
Acta Pharmacologica Sinica
Xi-shan Wu
Rui Wang
Yanli Xing
Xiaoqian Xue
Yan Zhang
Yong-Zhi Lu
Yu Song
Xiao-yu Luo
Chun Wu
Yulai Zhou
Jian-Qin Jiang
Yong Xu
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Citations (8)
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