Regioselective Synthesis of Indolopyrazines through a Sequential Rhodium-Catalyzed Formal [3 + 3] Cycloaddition and Aromatization Reaction of Diazoindolinimines with Azirines
2018
A regioselective synthetic method for the preparation of indolopyrazines was demonstrated through a sequential Rh-catalyzed formal [3+3] cycloaddition and aromatization reaction of a wide range of diazoindolinimines with azirines. Because the previously reported synthetic methods afforded mixtures of indolopyrazines, the present method using unsymmetrical azirines has a strong advantage from a regioselectivity viewpoint.
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