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Synthesis of BACE1 Inhibitors E2609/E2071 via Oxime–Olefin Cycloaddition Following a Process Risk Mitigation Strategy
Synthesis of BACE1 Inhibitors E2609/E2071 via Oxime–Olefin Cycloaddition Following a Process Risk Mitigation Strategy
2021
Dae-Shik Kim
Kazuhiro Yoshizawa
Branko Mitasev
Matthew J. Schnaderbeck
Huiming Zhang
Masayuki Omori
Akio Kayano
Mitsuo Nagai
Kazunori Wakasugi
Yuzo Watanabe
Farid Benayoud
Yuichi Suzuki
Takafumi Motoki
Toshihiko Kaneko
Mamoru Takaishi
Tasuku Ishida
Takeda Kunitoshi
Yoichi Kita
Noboru Yamamoto
Khan Afzal
Paschalis Dimopoulos
Christopher Neil Farthing
Adrian Hall
Arani Chanda
Lily Lu
Markus Bracke
Francis G. Fang
Keywords:
Combinatorial chemistry
Oxime
Olefin fiber
Cycloaddition
Chemistry
process
Risk management
Correction
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