Dearomatization of Indoles via Palladium-Catalyzed Allylic C–H Activation
2016
The first Pd-catalyzed allylic dearomatization of substituted indoles triggered by C–H bond activation is reported. The presence of a catalytic amount of 2,5-DMBQ is proven to be a key factor for the high yield. This one-pot tandem allylic C–H activation/dearomatization sequence provides a straightforward access to 3,3-disubstituted indolines.
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