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Laura Doyle
Laura Doyle
Novartis
Kinase
Biochemistry
Chemistry
In vitro
Cell
4
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97
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Design and synthesis of potent RSK inhibitors
2018
Bioorganic & Medicinal Chemistry Letters
Rama Jain
Michelle Mathur
Jiong Lan
Abran Costales
Gordana Atallah
Savithri Ramurthy
Sharadha Subramanian
Lina Setti
Paul Feucht
Bob Warne
Laura Doyle
Stephen E. Basham
Anne B. Jefferson
Brent A. Appleton
Mika Lindvall
Cynthia M. Shafer
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Citations (5)
Discovery of Potent and Selective RSK Inhibitors as Biological Probes.
2015
Journal of Medicinal Chemistry
Rama Jain
Michelle Mathur
Jiong Lan
Abran Costales
Gordana Atallah
Savithri Ramurthy
Sharadha Subramanian
Lina Setti
Paul Feucht
Bob Warne
Laura Doyle
Stephen E. Basham
Anne B. Jefferson
Mika Lindvall
Brent A. Appleton
Cynthia M. Shafer
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Citations (35)
Novel Potent and Selective Inhibitors of p90 Ribosomal S6 Kinase Reveal the Heterogeneity of RSK Function in MAPK- Driven Cancers
2014
Molecular Cancer Research
Ida Aronchik
Brent A. Appleton
Stephen E. Basham
Kenneth Crawford
Mercedita Del Rosario
Laura Doyle
William F. Estacio
Jiong Lan
Mika Lindvall
Catherine Luu
Elizabeth Ornelas
Eleni Venetsanakos
Cynthia M. Shafer
Anne B. Jefferson
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Citations (40)
2-Amino-7-substituted benzoxazole analogs as potent RSK2 inhibitors.
2014
Bioorganic & Medicinal Chemistry Letters
Abran Costales
Michelle Mathur
Savithri Ramurthy
Jiong Lan
Sharadha Subramanian
Rama Jain
Gordana Atallah
Lina Setti
Mika Lindvall
Brent A. Appleton
Elizabeth Ornelas
Paul Feucht
Bob Warne
Laura Doyle
Stephen E. Basham
Ida Aronchik
Anne B. Jefferson
Cynthia M. Shafer
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Citations (17)
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