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Kazuho Nakase
Kazuho Nakase
Merck & Co.
Biochemistry
Receptor
Chemistry
Antagonist
Radioligand
3
Papers
40
Citations
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Melanin-concentrating hormone 1-receptor antagonist suppresses body weight gain correlated with high receptor occupancy levels in diet-induced obesity mice
2009
European Journal of Pharmacology
Masahiko Ito
Akane Ishihara
Akira Gomori
Shinichiro Egashira
Hiroko Matsushita
Satoshi Mashiko
Junko Ito
Makoto Ito
Kazuho Nakase
Yuji Haga
Hisashi Iwaasa
Takao Suzuki
Norikazu Ohtake
Minoru Moriya
Nagaaki Sato
Douglas J. MacNeil
Norihiro Takenaga
Shigeru Tokita
Akio Kanatani
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Citations (18)
Discovery of novel diarylketoxime derivatives as selective and orally active melanin-concentrating hormone 1 receptor antagonists
2009
Bioorganic & Medicinal Chemistry Letters
Takao Suzuki
Minoru Kameda
Makoto Ando
Hiroshi Miyazoe
Etsuko Sekino
Satoru Ito
Kouta Masutani
Kaori Kamijo
Akihiro Takezawa
Minoru Moriya
Masahiko Ito
Junko Ito
Kazuho Nakase
Hiroko Matsushita
Akane Ishihara
Norihiro Takenaga
Shigeru Tokita
Akio Kanatani
Nagaaki Sato
Takehiro Fukami
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Citations (15)
Identification and characterization of a selective radioligand for melanin-concentrating hormone 1-receptor (MCH1R).
2009
Bioorganic & Medicinal Chemistry Letters
Masahiko Ito
Toshihiro Sakamoto
Takao Suzuki
Shinichiro Egashira
Minoru Moriya
Akane Ishihara
Hisashi Iwaasa
Hiroko Matsushita
Kazuho Nakase
Michael A. Wallace
Dennis C. Dean
Nagaaki Sato
Shigeru Tokita
Akio Kanatani
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Citations (7)
1