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Caroline Wetterstrand
Caroline Wetterstrand
Chemistry
Acetylcholine receptor
Allosteric modulator
Agonist
Allosteric regulation
4
Papers
158
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In vitro pharmacological profile of a novel α4β2 positive allosteric modulator NS9283 (A-969933)
2009
Biochemical Pharmacology
John Malysz
Tino Dyhring
Philip K. Ahring
Gunnar M. Olsen
Dan Peters
Jens Halvard Grønlien
Caroline Wetterstrand
Hilde Ween
M. Haakerud
Kirsten Thorin-Hagene
E. Andersen
David J. Anderson
Min Hu
Paul E. Kroeger
Chih-Hung Lee
Murali Gopalakrishnan
Daniel B. Timmermann
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Citations (6)
Discovery of 4-(5-(4-Chlorophenyl)-2-methyl-3-propionyl-1H-pyrrol-1-yl)benzenesulfonamide (A-867744) as a Novel Positive Allosteric Modulator of the α7 Nicotinic Acetylcholine Receptor
2009
Journal of Medicinal Chemistry
Ramin Faghih
Sujatha M. Gopalakrishnan
Jens Halvard Grønlien
John Malysz
Clark A. Briggs
Caroline Wetterstrand
Hilde Ween
Michael P. Curtis
Kathy Sarris
Gregory A. Gfesser
Rachid El Kouhen
Holly M. Robb
Richard J. Radek
Kennan C. Marsh
William H. Bunnelle
Murali Gopalakrishnan
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Citations (55)
In Vitro Pharmacological Characterization of a Novel Allosteric Modulator of α7 Neuronal Acetylcholine Receptor, 4-(5-(4-Chlorophenyl)-2-methyl-3-propionyl-1H-pyrrol-1-yl)benzenesulfonamide (A-867744), Exhibiting Unique Pharmacological Profile
2009
Journal of Pharmacology and Experimental Therapeutics
John Malysz
Jens Halvard Grønlien
David J. Anderson
Monika Håkerud
Kirsten Thorin-Hagene
Hilde Ween
Caroline Wetterstrand
Clark A. Briggs
Ramin Faghih
William H. Bunnelle
Murali Gopalakrishnan
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Citations (58)
Stimulation of dopamine release by nicotinic acetylcholine receptor ligands in rat brain slices correlates with the profile of high, but not low, sensitivity α4β2 subunit combination
2009
Biochemical Pharmacology
David J. Anderson
John Malysz
Jens Halvard Grønlien
Rachid El Kouhen
Monika Håkerud
Caroline Wetterstrand
Clark A. Briggs
Murali Gopalakrishnan
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Citations (39)
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