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Zhen-dong Chen
Zhen-dong Chen
Chinese Academy of Sciences
Pharmacology
Pharmacokinetics
Urine
Metabolite
Pharmacodynamics
5
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13
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Effects of Food on the Pharmacokinetic Properties and Mass Balance of Henagliflozin in Healthy Male Volunteers.
2021
Clinical Therapeutics
Zhen-dong Chen
Qian Chen
Yun-ting Zhu
Yifan Zhang
Yan Zhan
Xiao-Fei Chen
Xin Liang
Jingying Jia
Chen Yu
Hai-Yan Liu
Jian-Jun Zou
Yan-Mei Liu
Dafang Zhong
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Metabolite identification in preclinical and clinical phase of drug development.
2021
Current Drug Metabolism
Ya-li Wu
Lu-lu Pan
Zhen-dong Chen
Yuan-Dong Zheng
Xingxing Diao
Dafang Zhong
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Metabolic disposition of the EGFR covalent inhibitor furmonertinib in humans.
2021
Acta Pharmacologica Sinica
Jian Meng
Hua Zhang
Jing Jing Bao
Zhen-dong Chen
Xiao-yun Liu
Yifan Zhang
Yong Jiang
Liyan Miao
Dafang Zhong
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Furmonertinib (Alflutinib, AST2818) is a potential positive control drug comparable to rifampin for evaluation of CYP3A4 induction in sandwich-cultured primary human hepatocytes.
2021
Acta Pharmacologica Sinica
Ya-li Wu
Ya-ru Xue
Zitao Guo
Zhen-dong Chen
Xin-yu Ge
Dafang Zhong
Xingxing Diao
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Alflutinib (AST2818), primarily metabolized by CYP3A4, is a potent CYP3A4 inducer.
2020
Acta Pharmacologica Sinica
Xiao-yun Liu
Zitao Guo
Zhen-dong Chen
Yifan Zhang
Jialan Zhou
Yong Jiang
Qian-Yu Zhao
Xingxing Diao
Dafang Zhong
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Citations (9)
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