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Martin P. Schwalm
Martin P. Schwalm
Goethe University Frankfurt
Chemistry
Kinase
Small molecule
Cysteine
Cell biology
4
Papers
2
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0
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Discovery of a Potent and Highly Isoform-Selective Inhibitor of the Neglected Ribosomal Protein S6 Kinase Beta 2 (S6K2)
2021
ChemRxiv
Stefan Gerstenecker
Lisa Haarer
Martin Schröder
Mark Kudolo
Martin P. Schwalm
Valentin Wydra
Ricardo Augusto Massarico Serafim
Apirat Chaikuad
Stefan Knapp
Stefan Laufer
Matthias Gehringer
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Discovery of a Potent and Highly Isoform-Selective Inhibitor of the Neglected Ribosomal Protein S6 Kinase Beta 2 (S6K2).
2021
Cancers
Stefan Gerstenecker
Lisa Haarer
Martin Schröder
Mark Kudolo
Martin P. Schwalm
Valentin Wydra
Ricardo A. M. Serafim
Apirat Chaikuad
Stefan Knapp
Stefan Laufer
Matthias Gehringer
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Development of the First Covalent Monopolar Spindle Kinase 1 (MPS1/TTK) Inhibitor
2021
ChemRxiv
Ricardo A. M. Serafim
A.S. Santiago
Caio V dos Reis
J.E. Takarada
Priscila Mezzomo
Katlin B. Massirer
Martin P. Schwalm
Mark Kudolo
Stefan Gerstenecker
Apirat Chaikuad
Stefan Knapp
Stefan Laufer
Rafael M. Couñago
Matthias Gehringer
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Crystal Structure and Inhibitor Identifications Reveal Targeting Opportunity for the Atypical MAPK Kinase ERK3.
2020
International Journal of Molecular Sciences
Martin Schröder
Panagis Filippakopoulos
Martin P. Schwalm
Carla Alamillo Ferrer
David H. Drewry
Stefan Knapp
Apirat Chaikuad
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