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Juan Ge
Juan Ge
Hefei Institutes of Physical Science
Kinase
Biochemistry
Chemistry
In vivo
Cancer research
4
Papers
26
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0
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Discovery of (E)-N1-(3-fluorophenyl)-N3-(3-(2-(pyridin-2-yl)vinyl)-1H-indazol-6-yl)malonamide (CHMFL-KIT-033) as a Novel c-KIT T670I Mutant Selective Kinase Inhibitor for Gastrointestinal Stromal Tumors (GISTs)
2019
Journal of Medicinal Chemistry
Xuesong Liu
Beilei Wang
Cheng Chen
Ziping Qi
Fengming Zou
Junjie Wang
Chen Hu
Aoli Wang
Juan Ge
Qingwang Liu
Kailin Yu
Zhenquan Hu
Zongru Jiang
Wei Wang
Li Wang
Wenchao Wang
Tao Ren
Mingfeng Bai
Qingsong Liu
Jing Liu
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Citations (5)
Axitinib overcomes multiple imatinib resistant cKIT mutations including the gatekeeper mutation T670I in gastrointestinal stromal tumors
2019
Therapeutic Advances in Medical Oncology
Feiyang Liu
Fengming Zou
Cheng Chen
Kailin Yu
Xiaochuan Liu
Shuang Qi
Jiaxin Wu
Chen Hu
Zhenquan Hu
Juan Liu
Xuesong Liu
Li Wang
Juan Ge
Wenchao Wang
Tao Ren
Mingfeng Bai
Yujiao Cai
Xudong Xiao
Feng Qian
Jun Tang
Qingsong Liu
Jing Liu
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Discovery of 4-(((4-(5-chloro-2-(((1s,4s)-4-((2-methoxyethyl)amino)cyclohexyl)amino)pyridin-4-yl)thiazol-2-yl)amino)methyl)tetrahydro-2H-pyran-4-carbonitrile (JSH-150) as a novel highly selective and potent CDK9 kinase inhibitor
2018
European Journal of Medicinal Chemistry
Beilei Wang
Jiaxin Wu
Yun Wu
Cheng Chen
Fengming Zou
Aoli Wang
Hong Wu
Zhenquan Hu
Zongru Jiang
Qingwang Liu
Wei Wang
Yicong Zhang
Feiyang Liu
Ming Zhao
Jie Hu
Tao Huang
Juan Ge
Li Wang
Tao Ren
Yuxin Wang
Jing Liu
Qingsong Liu
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Citations (16)
Discovery of (S)-2-amino-N-(5-(6-chloro-5-(3-methylphenylsulfonamido)pyridin-3-yl)-4-methylthiazol-2-yl)-3-methylbutanamide (CHMFL-PI3KD-317) as a potent and selective phosphoinositide 3-kinase delta (PI3Kδ) inhibitor
2018
European Journal of Medicinal Chemistry
Xiaofei Liang
Feng Li
Cheng Chen
Zongru Jiang
Aoli Wang
Xiaochuan Liu
Juan Ge
Zhenquan Hu
Kailin Yu
Wenliang Wang
Fengming Zou
Qingwang Liu
Beilei Wang
Li Wang
Shanchun Zhang
Yuxin Wang
Qingsong Liu
Jing Liu
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