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Anil Desphande
Anil Desphande
University of Alabama at Birmingham
Potency
Tetralone
Organic chemistry
Biochemistry
Ligand (biochemistry)
2
Papers
29
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Methyl-substituted conformationally constrained rexinoid agonists for the retinoid X receptors demonstrate improved efficacy for cancer therapy and prevention.
2014
Bioorganic & Medicinal Chemistry
Anil Desphande
Gang Xia
LeeAnn J. Boerma
Kimberly K. Vines
Venkatram R. Atigadda
Susan M. Lobo-Ruppert
Clinton J. Grubbs
Fariba Moeinpour
Craig D. Smith
Konstantin Christov
Wayne J. Brouillette
Donald D. Muccio
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Citations (16)
Methyl substitution of a rexinoid agonist improves potency and reveals site of lipid toxicity.
2014
Journal of Medicinal Chemistry
Venkatram R. Atigadda
Gang Xia
Anil Desphande
LeeAnn J. Boerma
Susan M. Lobo-Ruppert
Clinton J. Grubbs
Craig D. Smith
Wayne J. Brouillette
Donald D. Muccio
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Citations (13)
1