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R. Curtis Haltiwanger
R. Curtis Haltiwanger
Cephalon
Chemistry
Stereochemistry
Combinatorial chemistry
Pharmacology
Antagonism
4
Papers
18
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3,4-Diaza-bicyclo[4.1.0]hept-4-en-2-one phenoxypropylamine analogs of irdabisant (CEP-26401) as potent histamine-3 receptor inverse agonists with robust wake-promoting activity
2015
European Journal of Medicinal Chemistry
Robert L. Hudkins
Nadine C. Becknell
Jacquelyn A. Lyons
Lisa D. Aimone
Mark Olsen
R. Curtis Haltiwanger
Joanne R. Mathiasen
Rita Raddatz
John A. Gruner
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Citations (9)
4-Phenoxypiperidine pyridazin-3-one histamine H3 receptor inverse agonists demonstrating potent and robust wake promoting activity
2012
Bioorganic & Medicinal Chemistry Letters
Robert L. Hudkins
Allison L. Zulli
Reddeppa reddy Dandu
Ming Tao
Kurt A. Josef
Lisa D. Aimone
R. Curtis Haltiwanger
Zeqi Huang
Jacquelyn A. Lyons
Joanne R. Mathiasen
Rita Raddatz
John A. Gruner
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Citations (9)
Novel forms a multi-cyclic compound
2010
Stephen Bierlmaier
Michael Christie
Laurent Courvoisier
R. Scott Field
R. Curtis Haltiwanger
Linli He
Martin J. Jacobs
Michael H. Kress
Robert E. Mckean
Dale R. Mowrey
Joseph Petraitis
Mehran Yazdanian
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Formes cristallines d'hydrochlorure de tiagabine
2007
Scott L. Childs
Leonard J. Chyall
Karen S. Gushurst
R. Curtis Haltiwanger
Robert E. Mckean
Donglai Yang
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