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Fei Jiang
Fei Jiang
China Pharmaceutical University
Chemistry
Biochemistry
BET inhibitor
BRD4
Small molecule
5
Papers
26
Citations
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Discovery of 1-(5-(1H-benzo[d]imidazole-2-yl)-2,4-dimethyl-1H-pyrrol-3-yl)ethan-1-one derivatives as novel and potent bromodomain and extra-terminal (BET) inhibitors with anticancer efficacy.
2022
European Journal of Medicinal Chemistry
Bo Kong
Zhaohong Zhu
Hongmei Li
Qianqian Hong
Cong Wang
Ma Yu
Wan Zheng
Fei Jiang
Zhimin Zhang
Ting Ran
Bian Yuanyuan
Na Yang
Tao Lu
Jiapeng Zhu
Weifang Tang
Yadong Chen
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The Discovery of Quinoline Derivatives, as NF-κB Inducing Kinase (NIK) Inhibitors with Anti-inflammatory Effects in Vitro, Low Toxicities against T Cell Growth
2020
Bioorganic & Medicinal Chemistry
Jianing Song
Yuqin Zhu
Weidong Zu
Chunqi Duan
Junyu Xu
Fei Jiang
Xinren Wang
Shuwen Li
Chenhe Liu
Qianqian Gao
Hongmei Li
Yanmin Zhang
Weifang Tang
Tao Lu
Yadong Chen
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Discovery of coumarin derivatives as potent and selective cyclin-dependent kinase 9 (CDK9) inhibitors with high antitumour activity
2020
European Journal of Medicinal Chemistry
Junyu Xu
Hongmei Li
Xinren Wang
Jianhang Huang
Shuwen Li
Chenhe Liu
Ruinan Dong
Gaoyuan Zhu
Chunqi Duan
Fei Jiang
Yanmin Zhang
Yuqin Zhu
Tianyi Zhang
Yadong Chen
Weifang Tang
Tao Lu
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Targeting BRD4 prevents acute gouty arthritis by regulating pyroptosis.
2020
International Journal of Biological Sciences
Kun Hao
Wenjiao Jiang
Mengze Zhou
Hanwen Li
Yadong Chen
Fei Jiang
Qing-Hua Hu
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Discovery of Novel Small Molecule Induced Selective Degradation of the Bromodomain and Extra-Terminal (BET) Bromodomain Protein BRD4 and BRD2 with Cellular Potencies
2019
Bioorganic & Medicinal Chemistry
Fei Jiang
Qingyun Wei
Huili Li
Hongmei Li
Yong Cui
Yu Ma
Haifang Chen
Peng Cao
Tao Lu
Yadong Chen
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Citations (12)
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