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Jun Sugama
Jun Sugama
Takeda Pharmaceutical Company
hERG
Somatostatin receptor
Chemistry
Somatostatin
Hormone
2
Papers
21
Citations
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Discovery of novel 5-oxa-2,6-diazaspiro[3.4]oct-6-ene derivatives as potent, selective, and orally available somatostatin receptor subtype 5 (SSTR5) antagonists for treatment of type 2 diabetes mellitus
2017
Bioorganic & Medicinal Chemistry
Hideki Hirose
Takeshi Yamasaki
Masaki Ogino
Ryo Mizojiri
Yumiko Tamura-Okano
Hiroaki Yashiro
Yo Muraki
Yoshihide Nakano
Jun Sugama
Akito Hata
Shinji Iwasaki
Masanori Watanabe
Tsuyoshi Maekawa
Shizuo Kasai
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Citations (14)
Discovery of novel somatostatin receptor subtype 5 (SSTR5) antagonists: Pharmacological studies and design to improve pharmacokinetic profiles and human Ether-a-go-go-related gene (hERG) inhibition
2017
Bioorganic & Medicinal Chemistry
Takeshi Yamasaki
Hideki Hirose
Tohru Yamashita
Nobuyuki Takakura
Sachie Morimoto
Takashi Nakahata
Asato Kina
Yoshihide Nakano
Yumiko Okano Tamura
Jun Sugama
Tomoyuki Odani
Yuji Shimizu
Shinji Iwasaki
Masanori Watanabe
Tsuyoshi Maekawa
Shizuo Kasai
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Citations (7)
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