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Richard Spring
Richard Spring
Schering-Plough
Chemistry
Melanin-concentrating hormone receptor
Organic chemistry
Structure–activity relationship
Piperidine
4
Papers
91
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Design and synthesis of orally efficacious piperidine-based melanin-concentrating hormone receptor 1 antagonists
2006
Bioorganic & Medicinal Chemistry Letters
Wen-Lian Wu
Duane A. Burnett
Mary Ann Caplen
Domalski
Chad E. Bennett
Richard Spring
Li Qiang
Thavalakulamgara K. Sasikumar
William J. Greenlee
Brian E. Hawes
Kim O’Neill
Blair Weig
Brian Spar
Daniel J. Weston
Timothy J. Kowalski
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Synthesis and structure–activity relationships of piperidine-based melanin-concentrating hormone receptor 1 antagonists
2006
Bioorganic & Medicinal Chemistry Letters
Wen-Lian Wu
Duane A. Burnett
Richard Spring
Li Qiang
Thavalakulamgara K. Sasikumar
Martin S. Domalski
William J. Greenlee
Kim O’Neill
Brian E. Hawes
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Citations (7)
Synthesis and structure–activity relationships of piperidine-based melanin-concentrating hormone receptor 1 antagonists
2006
Bioorganic & Medicinal Chemistry Letters
Wen-Lian Wu
Duane A. Burnett
Richard Spring
Li Qiang
Thavalakulamgara K. Sasikumar
Martin S. Domalski
William J. Greenlee
Kim O’Neill
Brian E. Hawes
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Citations (6)
Dopamine D1/D5 receptor antagonists with improved pharmacokinetics: Design, synthesis, and biological evaluation of phenol bioisosteric analogues of benzazepine D1/D5 antagonists
2005
Journal of Medicinal Chemistry
Wen-Lian Wu
Duane A. Burnett
Richard Spring
William J. Greenlee
Michelle Smith
Leonard Favreau
Ahmad Fawzi
Hongtao Zhang
Jean E. Lachowicz
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Citations (78)
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