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Koichi Yonezawa
Koichi Yonezawa
Astellas Pharma
Chemistry
Pharmacology
Neuropathic pain
CYP3A4
Biochemistry
5
Papers
87
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Synthesis, SAR study, and biological evaluation of novel 2,3-dihydro-1H-imidazo[1,2-a]benzimidazole derivatives as phosphodiesterase 10A inhibitors
2019
Bioorganic & Medicinal Chemistry
Ayaka Chino
Shugo Honda
Masataka Morita
Koichi Yonezawa
Wataru Hamaguchi
Yasushi Amano
Hiroyuki Moriguchi
Mayako Yamazaki
Masaki Aota
Masaki Tomishima
Naoyuki Masuda
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Citations (4)
Design, synthesis, and biological evaluation of novel biphenyl-4-carboxamide derivatives as orally available TRPV1 antagonists
2018
Bioorganic & Medicinal Chemistry
Hiromasa Oka
Koichi Yonezawa
Akio Kamikawa
Kazuhiro Ikegai
Norio Asai
Shohei Shirakami
Satoshi Miyamoto
Toshihiro Watanabe
Tetsuo Kiso
Yukihiro Takemoto
Seiji Tamura
Takahiro Kuramochi
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Discovery of an 8-methoxytetrahydroisoquinoline derivative as an orally active N-type calcium channel blocker for neuropathic pain without CYP inhibition liability
2015
Bioorganic & Medicinal Chemistry
Takashi Ogiyama
Koichi Yonezawa
Makoto Inoue
Naoko Katayama
Toshihiro Watanabe
Seiji Yoshimura
Takayasu Gotoh
Tetsuo Kiso
Akiko Koakutsu
Shuichiro Kakimoto
Jun-Ichi Shishikura
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Citations (4)
Discovery of a 1-isopropyltetrahydroisoquinoline derivative as an orally active N-type calcium channel blocker for neuropathic pain.
2015
Bioorganic & Medicinal Chemistry
Takashi Ogiyama
Koichi Yonezawa
Makoto Inoue
Toshihiro Watanabe
Yukihito Sugano
Takayasu Gotoh
Tetsuo Kiso
Akiko Koakutsu
Shuichiro Kakimoto
Jun-Ichi Shishikura
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Citations (6)
Amelioration of Neuropathic Pain by Novel Transient Receptor Potential Vanilloid 1 Antagonist AS1928370 in Rats without Hyperthermic Effect
2011
Journal of Pharmacology and Experimental Therapeutics
Tomonari Watabiki
Tetsuo Kiso
Takahiro Kuramochi
Koichi Yonezawa
Noriko Tsuji
Atsuyuki Kohara
Shuichiro Kakimoto
Toshiaki Aoki
Nobuya Matsuoka
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Citations (72)
1