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David Spalding
David Spalding
University of Hertfordshire
Biochemistry
Chemistry
In vitro
Selectivity
Antagonist
2
Papers
109
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The discovery of 6-[2-(5-chloro-2-{[(2,4-difluorophenyl)methyl]oxy}phenyl)-1-cyclopenten-1-yl]-2-pyridinecarboxylic acid, GW848687X, a potent and selective prostaglandin EP1 receptor antagonist for the treatment of inflammatory pain
2007
Bioorganic & Medicinal Chemistry Letters
Gerard Martin Paul Giblin
Rino A. Bit
Susan H. Brown
Helene M. Chaignot
Anita Chowdhury
Iain P. Chessell
Nicholas Maughan Clayton
Tanya Coleman
Adrian Hall
Beverley Hammond
David Nigel Hurst
Anton D. Michel
Alan Naylor
Riccardo Novelli
Tiziana Scoccitti
David Spalding
Sac P. Tang
Alex W. Wilson
Rich Wilson
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Citations (42)
Indazolylamino quinazolines and pyridopyrimidines as inhibitors of the EGFr and c-erbB-2
2001
Bioorganic & Medicinal Chemistry Letters
Stuart Cockerill
Colin Stubberfield
Jeremy Stables
Malcolm Clive Carter
Stephen Guntrip
Kathryn J. GlaxoSmithKline Smith
Steve McKeown
Robert Shaw
Peter Topley
Lindy Thomsen
Karen Affleck
Amanda Jowett
David J. Hayes
Malcolm Willson
Patrick Woollard
David Spalding
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Citations (67)
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