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Yoshiyuki Tenda
Yoshiyuki Tenda
Adenosine
Ligand (biochemistry)
Adenosine A1 receptor
Biochemistry
Chemistry
3
Papers
90
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Design, Synthesis and Biological Evaluation of a Novel Series of Potent, Orally Active Adenosine A1 Receptor Antagonists with High Blood-Brain Barrier Permeability
2001
Chemical & Pharmaceutical Bulletin
Satoru Kuroda
Fujiko Takamura
Yoshiyuki Tenda
Hiromichi Itani
Yasuyo Tomishima
Atsushi Akahane
Kazuo Sakane
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Citations (24)
Novel adenosine A1 receptor antagonists. Synthesis and structure-activity relationships of a novel series of 3-(2-cyclohexenyl-3-oxo-2,3-dihydropyridazin-6-yl)-2-phenylpyrazolo[1,5 -a]pyridines.
2000
Bioorganic & Medicinal Chemistry
Satoru Kuroda
Atsushi Akahane
Hiromichi Itani
Shintaro Nishimura
Kieran Durkin
Yoshiyuki Tenda
Kazuo Sakane
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Citations (25)
Discovery of FR166124, a novel water-soluble pyrazolo-[1,5-α]pyridine adenosine A1 receptor antagonist
1999
Bioorganic & Medicinal Chemistry Letters
Satoru Kuroda
Atsushi Akahane
Hiromichi Itani
Shintaro Nishimura
Kieran Durkin
Takayoshi Kinoshita
Yoshiyuki Tenda
Kazuo Sakane
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Citations (41)
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