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Stéphane A.H. Spieser
Stéphane A.H. Spieser
Merck & Co.
Chemistry
Photochemistry
Dimethyldioxirane
Regioselectivity
Bicyclic molecule
4
Papers
43
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Regioselective Synthesis of 7,8-Dihydropyrrolo[1,2-a]pyrimidin-4(6H)-ones and 7,8-Dihydropyrrolo[1,2-α]pyrimidin-2(6H)-ones
2010
Synlett
Monica Donghi
Silvia Pesci
Vincenzo Summa
Uwe Koch
Stéphane A.H. Spieser
Cristina Gardelli
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Regioselective Synthesis of7,8-Dihydropyrrolo[1,2-a]pyrimidin-4(6H)-ones and 7,8-Dihydropyrrolo[1,2-a]pyrimidin-2(6H)-ones
2010
Synlett
Monica Donghi
Silvia Pesci
Vincenzo Summa
Uwe Koch
Stéphane A.H. Spieser
Cristina Gardelli
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Dihydroxy-pyrimidine and N-methylpyrimidone HIV-integrase inhibitors: Improving cell based activity by the quaternarization of a chiral center
2009
Bioorganic & Medicinal Chemistry Letters
Emanuela Nizi
Maria Vittoria Orsale
Benedetta Crescenzi
Giovanna Pescatore
Ester Muraglia
Anna Alfieri
Cristina Gardelli
Stéphane A.H. Spieser
Vincenzo Summa
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Citations (11)
4-Hydroxy-5-pyrrolinone-3-carboxamide HIV-1 integrase inhibitors
2008
Bioorganic & Medicinal Chemistry Letters
Paola Pace
Stéphane A.H. Spieser
Vincenzo Summa
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Citations (32)
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