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Eugene Kelleher
Eugene Kelleher
Chemistry
Stereochemistry
Medicinal chemistry
Protein kinase B
Structure–activity relationship
4
Papers
42
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Discovery of 3-(3-(4-(1-Aminocyclobutyl)phenyl)-5-phenyl-3H-imidazo[4,5-b]pyridin-2-yl)pyridin-2-amine (ARQ 092): An Orally Bioavailable, Selective, and Potent Allosteric AKT Inhibitor
2016
Journal of Medicinal Chemistry
Jean-Marc Lapierre
Sudharshan Eathiraj
David Vensel
Yanbin Liu
Cathy Bull
Susan Cornell-Kennon
Shin Iimura
Eugene Kelleher
Darin Kizer
Steffi Koerner
Sapna Makhija
Akihisa Matsuda
Magdi Moussa
Nivedita Namdev
Ronald E. Savage
Jeff Szwaya
Erika Volckova
Neil Westlund
Hui Wu
Brian S. Schwartz
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Citations (42)
Composés de benzo-pyrido-triazolo-diazépine substitués
2011
Syed M. Ali
Mark A. Ashwell
Eugene Kelleher
Steffi Koerner
Jean-Marc Lapierre
Jeffrey S. Link
Yanbin Liu
Magdi Moussa
Rocio Palma
Manish Tandon
David Vensel
Neil Westlund
Hui Wu
Rui-Yang Yang
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Composés de 5,6-dihydro-6-phénylbenzo[f]isoquinoléine-2-amines substituées
2009
Syed M. Ali
Mark A. Ashwell
Manish Tandon
Rui-Yang Yang
Yanbin Liu
David Vensel
Sudharshan Eathiraj
Rocio Palma
Jean-Marc Lapierre
Neil Westlund
Hui Wu
Nivedita Namdev
Eugene Kelleher
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Dérivés de pyrrolidinone, pyrrolidine-2,5-dione, pyrrolidine et thiosuccinimide, compositions et procédés pour le traitement d'un cancer
2008
Jianqiang Wang
Syed M. Ali
Eugene Kelleher
Yanbin Liu
Jason Hill
Mark A. Ashwell
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