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Haruka Imada
Haruka Imada
Takeda Pharmaceutical Company
Phosphodiesterase
Biochemistry
Chemistry
Pharmacology
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4
Papers
56
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The phosphodiesterase 2A inhibitor TAK-915 ameliorates cognitive impairments and social withdrawal in N-methyl-D-aspartate receptor antagonist-induced rat models of schizophrenia
2018
Journal of Pharmacology and Experimental Therapeutics
Masato Nakashima
Haruka Imada
Eri Shiraishi
Yuki Ito
Noriko Suzuki
Maki Miyamoto
Takahiko Taniguchi
Hiroki Iwashita
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Citations (13)
T257. The Phosphodiesterase 2A Inhibitor TAK-915 Ameliorates Cognitive Impairments and Social Withdrawal in N-Methyl-D-Aspartate Receptor Antagonist-Induced Rat Models of Schizophrenia
2018
Biological Psychiatry
Masato Nakashima
Haruka Imada
Eri Shiraishi
Yuki Ito
Noriko Suzuki
Maki Miyamoto
Takahiko Taniguchi
Hiroki Iwashita
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Discovery of an Orally Bioavailable, Brain-Penetrating, in Vivo Active Phosphodiesterase 2A Inhibitor Lead Series for the Treatment of Cognitive Disorders
2017
Journal of Medicinal Chemistry
Satoshi Mikami
Shigekazu Sasaki
Yasutomi Asano
Osamu Ujikawa
Shoji Fukumoto
Kosuke Nakashima
Hideyuki Oki
Naomi Kamiguchi
Haruka Imada
Hiroki Iwashita
Takahiko Taniguchi
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Citations (21)
Discovery of Clinical Candidate N-((1S)-1-(3-Fluoro-4-(trifluoromethoxy)phenyl)-2-methoxyethyl)-7-methoxy-2-oxo-2,3-dihydropyrido[2,3-b]pyrazine-4(1H)-carboxamide (TAK-915): A Highly Potent, Selective, and Brain-Penetrating Phosphodiesterase 2A Inhibitor for the Treatment of Cognitive Disorders.
2017
Journal of Medicinal Chemistry
Satoshi Mikami
Shinji Nakamura
Tomoko Ashizawa
Izumi Nomura
Masanori Kawasaki
Shigekazu Sasaki
Hideyuki Oki
Hironori Kokubo
Isaac D. Hoffman
Hua Zou
Noriko Uchiyama
Kosuke Nakashima
Naomi Kamiguchi
Haruka Imada
Noriko Suzuki
Hiroki Iwashita
Takahiko Taniguchi
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Citations (21)
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