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Margaret L. Gregory
Margaret L. Gregory
Pfizer
Testosterone
Antagonist
Chemistry
Gonadotropin-releasing hormone
Biochemistry
4
Papers
97
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Discovery of a novel, orally active, small molecule gonadotropin-releasing hormone (GnRH) receptor antagonist
2006
Journal of Medicinal Chemistry
Haitao Li
Kenna Anderes
Eugenia Kraynov
David Robert Luthin
Quyen-Quyen T. Do
Yufeng Hong
Eileen Valenzuela Tompkins
Eric T. Sun
Ranjan Jagath Rajapakse
Ved P. Pathak
Lance Christopher Christie
Haresh Vazir
Rosemary Castillo
Margaret L. Gregory
Mary Castro
Karen Nared-Hood
and Genevieve Paderes
Mark B. Anderson
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Citations (17)
Biological Characterization of a Novel, Orally Active Small Molecule Gonadotropin-Releasing Hormone (GnRH) Antagonist Using Castrated and Intact Rats
2003
Journal of Pharmacology and Experimental Therapeutics
Kenna Anderes
David Robert Luthin
Rosemary Castillo
Eugenia Kraynov
Mary Castro
Karen Nared-Hood
Margaret L. Gregory
Ved P. Pathak
Lance Christopher Christie
Genevieve Paderes
Haresh Vazir
Qiang Ye
Mark B. Anderson
John May
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Citations (47)
Effect of Testosterone Suppression on the Pharmacokinetics of a Potent GnRH Receptor Antagonist
2002
Pharmaceutical Research
Eugenia A. Iatsimirskaia
Margaret L. Gregory
Kenna Anderes
Rosemary Castillo
K. Eric Milgram
David R. Luthin
Ved P. Pathak
Lance Christopher Christie
Haresh Vazir
Mark B. Anderson
John May
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Citations (9)
Characterization of mono- and diaminopyrimidine derivatives as novel, nonpeptide gonadotropin releasing hormone (GnRH) receptor antagonists
2002
Bioorganic & Medicinal Chemistry Letters
David R. Luthin
Yufeng Hong
Eileen Valenzuela Tompkins
Kenna Anderes
Genevieve Paderes
Eugenia Kraynov
Mary Castro
Karen Nared-Hood
Rosemary Castillo
Margaret L. Gregory
Haresh Vazir
John May
Mark B. Anderson
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Citations (24)
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