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Keisuke Kashimoto
Keisuke Kashimoto
Kyoto Pharmaceutical University
Peptidomimetic
Plasmepsin
Chemistry
Stereochemistry
Malaria
3
Papers
18
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Optimization of plasmepsin inhibitor by focusing on similar structural feature with chloroquine to avoid drug-resistant mechanism of Plasmodium falciparum
2014
Bioorganic & Medicinal Chemistry Letters
Takuya Miura
Koushi Hidaka
Yukiko Azai
Keisuke Kashimoto
Yuko Kawasaki
Shen En Chen
Renato F. Freitas
Ernesto Freire
Yoshiaki Kiso
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Optimization of Peptidomimetic Plasmepsin Inhibitor Containing Allophenylnorstatine Using Basic Substituent for Malaria Treatment
2011
Takuya Miura
Koushi Hidaka
Keisuke Kashimoto
Yuto Hori
Yukiko Azai
Yuko Kawasaki
J Ruben Adam
Ernesto Freire
Tooru Kimura
Yoshiaki Kiso
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Improvement of both plasmepsin inhibitory activity and antimalarial activity by 2-aminoethylamino substitution
2010
Bioorganic & Medicinal Chemistry Letters
Takuya Miura
Koushi Hidaka
Tsuyoshi Uemura
Keisuke Kashimoto
Yuto Hori
Yuko Kawasaki
Adam J. Ruben
Ernesto Freire
Tooru Kimura
Yoshiaki Kiso
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Citations (14)
1