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Youichi Nishikawa
Youichi Nishikawa
Takeda Pharmaceutical Company
CCR5 receptor antagonist
Biochemistry
Chemistry
Stereochemistry
Chemical synthesis
4
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278
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Discovery of a piperidine-4-carboxamide CCR5 antagonist (TAK-220) with highly potent Anti-HIV-1 activity.
2006
Journal of Medicinal Chemistry
Shinichi Imamura
Takashi Ichikawa
Youichi Nishikawa
Naoyuki Kanzaki
Katsunori Takashima
Shin-Ichi Niwa
Yuji Iizawa
Masanori Baba
Yoshihiro Sugihara
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Citations (59)
CCR5 antagonists as anti-HIV-1 agents. Part 3: Synthesis and biological evaluation of piperidine-4-carboxamide derivatives
2005
Bioorganic & Medicinal Chemistry
Shinichi Imamura
Youichi Nishikawa
Takashi Ichikawa
Taeko Hattori
Yoshihiro Matsushita
Shohei Hashiguchi
Naoyuki Kanzaki
Yuji Iizawa
Masanori Baba
Yoshihiro Sugihara
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Citations (41)
CCR5 antagonists as anti-HIV-1 agents. Part 2: Synthesis and biological evaluation of N-[3-(4-benzylpiperidin-1-yl)propyl]-N,N′-diphenylureas
2004
Bioorganic & Medicinal Chemistry
Shinichi Imamura
Osamu Kurasawa
Yoshi Nara
Takashi Ichikawa
Youichi Nishikawa
Takehiro Iida
Shohei Hashiguchi
Naoyuki Kanzaki
Yuji Iizawa
Masanori Baba
Yoshihiro Sugihara
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Citations (16)
Discovery of Novel, Potent, and Selective Small-Molecule CCR5 Antagonists as Anti-HIV-1 Agents: Synthesis and Biological Evaluation of Anilide Derivatives with a Quaternary Ammonium Moiety
2000
Journal of Medicinal Chemistry
Mitsuru Shiraishi
Yoshio Aramaki
Masaki Seto
Hiroshi Imoto
Youichi Nishikawa
Naoyuki Kanzaki
Mika Okamoto
Hidekazu Sawada
Osamu Nishimura
and Masanori Baba
Masahiko Fujino
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Citations (162)
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