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Hiroaki Oguri
Hiroaki Oguri
Gifu Pharmaceutical University
Reductase
Chemistry
Prostate cancer
castration resistant
Biochemistry
5
Papers
30
Citations
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2024
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Development ofNovel AKR1C3 Inhibitors as New PotentialTreatment for Castration-Resistant Prostate Cancer
2020
Journal of Medicinal Chemistry
Satoshi Endo
Hiroaki Oguri
Jin Segawa
Mina Kawai
Dawei Hu
Shuang Xia
Takuya Okada
Katsumasa Irie
Shinya Fujii
Hiroaki Gouda
Kazuhiro Iguchi
Takuo Matsukawa
Naohiro Fujimoto
Toshiyuki Nakayama
Naoki Toyooka
Toshiyuki Matsunaga
Akira Ikari
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Development of novel AKR1C3 inhibitors as new potential treatment for castration-resistant prostate cancer.
2020
Journal of Medicinal Chemistry
Satoshi Endo
Hiroaki Oguri
Jin Segawa
Mina Kawai
Dawei Hu
Shuang Xia
Takuya Okada
Katsumasa Irie
Shinya Fujii
Hiroaki Gouda
Kazuhiro Iguchi
Takuo Matsukawa
Naohiro Fujimoto
Toshiyuki Nakayama
Naoki Toyooka
Toshiyuki Matsunaga
Akira Ikari
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Citations (8)
Development and characterization of novel AKR1C3 inhibitors: Therapeutic potential for castration-resistant prostate cancer
2019
European Urology Supplements
N. Fujimoto
Satoshi Endo
Hiroaki Oguri
Naoki Toyooka
Toshiyuki Matsunaga
Akira Ikari
I. Tomisaki
T. Nakayama
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Synthesis of Potent and Selective Inhibitors of Aldo-Keto Reductase 1B10 and Their Efficacy against Proliferation, Metastasis, and Cisplatin Resistance of Lung Cancer Cells
2017
Journal of Medicinal Chemistry
Satoshi Endo
Shuang Xia
Miho Suyama
Yoshifumi Morikawa
Hiroaki Oguri
Dawei Hu
Yoshinori Ao
Satoyuki Takahara
Yoshikazu Horino
Yoshihiro Hayakawa
Yurie Watanabe
Hiroaki Gouda
Akira Hara
Kazuo Kuwata
Naoki Toyooka
Toshiyuki Matsunaga
Akira Ikari
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Citations (12)
Synthesis of 8-hydroxy-2-iminochromene derivatives as selective and potent inhibitors of human carbonyl reductase 1
2015
Organic and Biomolecular Chemistry
Dawei Hu
Namiki Miyagi
Yuki Arai
Hiroaki Oguri
Takeshi Miura
Toru Nishinaka
Tomoyuki Terada
Hiroaki Gouda
Ossama El-Kabbani
Shuang Xia
Naoki Toyooka
Akira Hara
Toshiyuki Matsunaga
Akira Ikari
Satoshi Endo
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Citations (10)
1