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Farhana Barmare
Farhana Barmare
Vertex Pharmaceuticals
CCR2
CCL2
Chemokine
Receptor
Chemistry
2
Papers
69
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When structure-affinity relationships meet structure-kinetics relationships: 3-((Inden-1-yl)amino)-1-isopropyl-cyclopentane-1-carboxamides as CCR2 antagonists.
2015
European Journal of Medicinal Chemistry
Maris Vilums
Annelien J.M. Zweemer
Farhana Barmare
Anouk M.F. van der Gracht
Dave C.T. Bleeker
Zhiyi Yu
Henk de Vries
Raymond S. Gross
Jeremy Clemens
Paul Krenitsky
Johannes Brussee
Dean Stamos
John Saunders
Laura H. Heitman
Adriaan P. IJzerman
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Citations (18)
Structure-kinetic relationships--an overlooked parameter in hit-to-lead optimization: a case of cyclopentylamines as chemokine receptor 2 antagonists.
2013
Journal of Medicinal Chemistry
Maris Vilums
Annelien J.M. Zweemer
Zhiyi Yu
Henk de Vries
Julia M. Hillger
Hannah Wapenaar
Ilse A. E. Bollen
Farhana Barmare
Raymond S. Gross
Jeremy Clemens
Paul Krenitsky
Johannes Brussee
Dean Stamos
John Saunders
Laura H. Heitman
Adriaan P. IJzerman
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Citations (51)
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