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Tatsuo Akaki
Tatsuo Akaki
Japan Tobacco
Stereochemistry
Pyruvate dehydrogenase complex
Chemistry
Ligand efficiency
Binding site
2
Papers
1
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0
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Structure-based drug design of novel and highly potent pyruvate dehydrogenase kinase inhibitors
2021
Bioorganic & Medicinal Chemistry
Yuki Bessho
Tatsuo Akaki
Yoshinori Hara
Maki Yamakawa
Shingo Obika
Genki Mori
Minoru Ubukata
Katsutaka Yasue
Yoshitomi Nakane
Yasuo Terasako
Takuya Orita
Satoki Doi
Tomoko Iwanaga
Ayumi Fujishima
Tsuyoshi Adachi
Hiroshi Ueno
Takahisa Motomura
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Fragment-based lead discovery to identify novel inhibitors that target the ATP binding site of pyruvate dehydrogenase kinases
2021
Bioorganic & Medicinal Chemistry
Tatsuo Akaki
Yuki Bessho
Takashi Ito
Fujioka Shingo
Minoru Ubukata
Genki Mori
Kenji Yamanaka
Takuya Orita
Satoki Doi
Tomoko Iwanaga
Kazutaka Ikegashira
Yoshiji Hantani
Isao Nakanishi
Tsuyoshi Adachi
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