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Xin Xue
Xin Xue
China Pharmaceutical University
Chemistry
Biochemistry
Stereochemistry
Potency
Luciferase
5
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95
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Novel IKKβ inhibitors discovery based on the co-crystal structure by using binding-conformation-based and ligand-based method.
2013
European Journal of Medicinal Chemistry
Jing-Jie Huang
Xiaowen Wu
Jian-Min Jia
Xiaoke Guo
Xin Xue
Zhengyu Jiang
Shenglie Zhang
Xiaojin Zhang
Haopeng Sun
Qidong You
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Citations (7)
3-aroylmethylene-2,3,6,7-tetrahydro-1H-pyrazino[2,1-a]isoquinolin-4(11bH)-ones as potent Nrf2/ARE inducers in human cancer cells and AOM-DSS treated mice.
2013
Journal of Medicinal Chemistry
Mei-Yang Xi
Jian-Min Jia
Haopeng Sun
Zhongying Sun
Jie-wei Jiang
Yajing Wang
Min-ye Zhang
Jun-Feng Zhu
Li-Li Xu
Zheng-Yu Jiang
Xin Xue
Ming Ye
Xi Yang
Yuan Gao
Lei Tao
Xiaoke Guo
Xiao-Li Xu
Qinglong Guo
Xiaojin Zhang
Rong Hu
Qidong You
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Citations (34)
Synthesis and bioevaluation of a series of α-pyrone derivatives as potent activators of Nrf2/ARE pathway (part I).
2013
European Journal of Medicinal Chemistry
Mei-Yang Xi
Zhongying Sun
Haopeng Sun
Jian-Min Jia
Zhengyu Jiang
Lei Tao
Ming Ye
Xi Yang
Yajing Wang
Xin Xue
Jing-Jie Huang
Yuan Gao
Xiaoke Guo
Shenglie Zhang
Yingrui Yang
Qinglong Guo
Rong Hu
Qidong You
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Citations (24)
Effective Screening Strategy Using Ensembled Pharmacophore Models Combined with Cascade Docking: Application to p53-MDM2 Interaction Inhibitors
2013
Journal of Chemical Information and Modeling
Xin Xue
Jinlian Wei
Li-Li Xu
Mei-Yang Xi
Xiao-Li Xu
Fang Liu
Xiaoke Guo
Lei Wang
Xiaojin Zhang
Ming-Ye Zhang
Meng-Chen Lu
Haopeng Sun
Qidong You
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Citations (22)
Studies on Chemical Structure Modification and StructureActivity Relationship of Derivatives of Gambogic Acid at C(39)
2012
Chemistry & Biodiversity
Haopeng Sun
Zongliang Liu
Xin Xue
Yuan Gao
Lei Zhang
Jinxin Wang
Qinglong Guo
Qidong You
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Citations (8)
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