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Yuji Nishiura
Yuji Nishiura
Biochemistry
Chemistry
In vivo
Benzimidazole
Ligand (biochemistry)
4
Papers
51
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Discovery of a novel olefin derivative as a highly potent and selective acetyl-CoA carboxylase 2 inhibitor with in vivo efficacy
2018
Bioorganic & Medicinal Chemistry Letters
Yuji Nishiura
Akira Matsumura
Naotake Kobayashi
Atsuyuki Shimazaki
Shingo Sakamoto
Naohisa Kitade
Yutaka Tonomura
Akira Ino
Takayuki Okuno
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Citations (9)
Identification of a novel benzimidazole derivative as a highly potent NPY Y5 receptor antagonist with an anti-obesity profile.
2013
Bioorganic & Medicinal Chemistry Letters
Yuusuke Tamura
Kyouhei Hayashi
Naoki Omori
Yuji Nishiura
Kana Watanabe
Nobuyuki Tanaka
Masahiko Fujioka
Naoki Kouyama
Akira Yukimasa
Yukari Tanaka
Takeshi Chiba
Hideki Tanioka
Hirohide Nambu
Hideo Yukioka
Hiroki Sato
Takayuki Okuno
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Citations (6)
Identification of a novel and orally available benzimidazole derivative as an NPY Y5 receptor antagonist with in vivo efficacy
2012
Bioorganic & Medicinal Chemistry Letters
Yuusuke Tamura
Naoki Omori
Naoki Kouyama
Yuji Nishiura
Kyouhei Hayashi
Kana Watanabe
Yukari Tanaka
Takeshi Chiba
Hideo Yukioka
Hiroki Sato
Takayuki Okuno
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Citations (13)
Design, synthesis and identification of novel benzimidazole derivatives as highly potent NPY Y5 receptor antagonists with attractive in vitro ADME profiles
2012
Bioorganic & Medicinal Chemistry Letters
Yuusuke Tamura
Naoki Omori
Naoki Kouyama
Yuji Nishiura
Kyouhei Hayashi
Kana Watanabe
Yukari Tanaka
Takeshi Chiba
Hideo Yukioka
Hiroki Sato
Takayuki Okuno
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Citations (23)
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