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Susan M Cusick
Susan M Cusick
Prodrug
Chemistry
In vivo
Ceftibuten
ED50
2
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3
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0
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2024
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Microbiological characterization of VNRX-5236: a broad spectrum β-lactamase inhibitor for rescue of the orally bioavailable cephalosporin ceftibuten as a carbapenem-sparing agent against strains of Enterobacterales expressing extended spectrum β-lactamases and serine carbapenemases.
2021
Antimicrobial Agents and Chemotherapy
Cassandra L Chatwin
Hamrick Jodie
Robert E. Lee Trout
Cullen L. Myers
Susan M Cusick
William J. Weiss
Mark Pulse
Luigi Xerri
Christopher J. Burns
Gregory Moeck
Denis M. Daigle
Kaitlyn John
Tsuyoshi Uehara
Daniel C. Pevear
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Citations (2)
Discovery of VNRX-7145 (VNRX-5236 Etzadroxil): An Orally Bioavailable β-Lactamase Inhibitor for Enterobacterales Expressing Ambler Class A, C, and D Enzymes.
2021
Journal of Medicinal Chemistry
Robert E. Lee Trout
Allison L. Zulli
Eugen F. Mesaros
Randy W. Jackson
Boyd Steven A
Bin Liu
Jodie Hamrick
Denis M. Daigle
Cassandra L Chatwin
Kaitlyn John
Lisa McLaughlin
Susan M Cusick
William J. Weiss
Mark Pulse
Daniel C. Pevear
Greg Moeck
Luigi Xerri
Christopher J. Burns
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Citations (1)
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