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Karen A. Tricarico
Karen A. Tricarico
Biochemistry
Renin–angiotensin system
Renin inhibitor
Chemistry
Enzyme
4
Papers
90
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Studies directed toward the design of orally active renin inhibitors. 2. Development of the efficacious, bioavailable renin inhibitor (2S)-2-benzyl-3-[[(1-methylpiperazin-4-yl)sulfonyl]propionyl]-3-thiazol-4-yl-L- alanine amide of (2S,3R,4S)-2-amino-1-cyclohexyl-3,4-dihydroxy-6-methylheptane (A-72517)
1993
Journal of Medicinal Chemistry
Saul H. Rosenberg
Kenneth P. Spina
Stephen L. Condon
Jim Polakowski
Zhengli Yao
Peter Kovar
Herman H. Stein
Jerome Cohen
Jennifer L. Barlow
Vered Klinghofer
David A. Egan
Karen A. Tricarico
Thomas J. Perun
William R. Baker
Hollis D. Kleinert
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Citations (41)
Design of a well-absorbed renin inhibitor
1991
Journal of Medicinal Chemistry
Saul H. Rosenberg
Hollis D. Kleinert
Herman H. Stein
Donald L. Martin
Marcia A. Chekal
Jerome Cohen
David A. Egan
Karen A. Tricarico
William R. Baker
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Citations (34)
Biochemical and pharmacological properties of ABBOTT-65317, a potent renin inhibitor
1990
European Journal of Pharmacology
Herman H. Stein
Saul H. Rosenberg
Jerome Cohen
Keith W. Woods
Donald L. Martin
Gary A. Young
James S. Polakowski
Patrick A. Marcotte
Karen A. Tricarico
Jacob J. Plattner
H.D. Kleinen
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Citations (1)
Human placental chorionic renin: production, purification and characterization
1988
Biochimica et Biophysica Acta
David A. Egan
Valerie Grzegorczyk
Karen A. Tricarico
Annemarie Rueter
William H. Holleman
Patrick Marcotte
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Citations (14)
1