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Shuyuan Zhao
Shuyuan Zhao
Janssen Pharmaceutica
Biochemistry
Agonist
Free fatty acid receptor 1
Pharmacology
In vivo
4
Papers
30
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Discovery of a Novel Potent GPR40 Full Agonist
2018
Bioorganic & Medicinal Chemistry Letters
Sanath K. Meegalla
Hui Huang
Tonya Martin
June Xu
Shuyuan Zhao
Jianying Liu
Meghan Hall
Joe Gunnet
Yuanping Wang
Brian Rady
Jose Silva
Monicah Otieno
Eric Arnoult
S. Paul Lee
Alessandro Pocai
Mark R. Player
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Citations (5)
GPR40-Mediated Gα12 Activation by Allosteric Full Agonists Highly Efficacious at Potentiating Glucose-Stimulated Insulin Secretion in Human Islets
2018
Molecular Pharmacology
Marie-Laure Rives
Brian Rady
Nadia Swanson
Shuyuan Zhao
Jenson Qi
Eric Arnoult
Ivona Bakaj
Arturo Mancini
Billy Breton
Paul S. Lee
Mark R. Player
Alessandro Pocai
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Citations (12)
6-Benzhydryl-4-amino-quinolin-2-ones as Potent Cannabinoid Type 1 (CB1) Receptor Inverse Agonists and Chemical Modifications for Peripheral Selectivity
2018
Journal of Medicinal Chemistry
Yue-Mei Zhang
Michael N. Greco
Mark J. Macielag
Christopher A. Teleha
Renee L. DesJarlais
Yuting Tang
George Ho
Cuifen Hou
Cailin Chen
Shuyuan Zhao
Jack Kauffman
Raul Camacho
Jenson Qi
William V. Murray
Keith T. Demarest
James Leonard
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Citations (10)
Discovery of novel benzo[b]thiophene tetrazoles as non-carboxylate GPR40 agonists
2017
Bioorganic & Medicinal Chemistry Letters
Hui Huang
Michael P. Winters
Sanath K. Meegalla
Eric Arnoult
S. Paul Lee
Shuyuan Zhao
Tonya Martin
Brian Rady
Jianying Liu
Meghan Towers
Monicah Otieno
Fran Xu
Heng Keang Lim
Jose Silva
Alessandro Pocai
Mark R. Player
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Citations (3)
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