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Toshiya Harasawa
Toshiya Harasawa
Takeda Pharmaceutical Company
Agonist
Chemistry
Dopamine receptor D2
Receptor
Pharmacology
3
Papers
51
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Design and synthesis of 1-(1-benzothiophen-7-yl)-1 H -pyrazole, a novel series of G protein-coupled receptor 52 (GPR52) agonists
2018
Bioorganic & Medicinal Chemistry
Takashi Nakahata
Kazuyuki Tokumaru
Yoshiteru Ito
Naoki Ishii
Masaki Setoh
Yuji Shimizu
Toshiya Harasawa
Kazunobu Aoyama
Teruki Hamada
Masakuni Kori
Kazuyoshi Aso
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Citations (9)
FTBMT, a Novel and Selective GPR52 Agonist, Demonstrates Antipsychotic-Like and Procognitive Effects in Rodents, Revealing a Potential Therapeutic Agent for Schizophrenia
2017
Journal of Pharmacology and Experimental Therapeutics
Keiji Nishiyama
Hirobumi Suzuki
Toshiya Harasawa
Noriko Suzuki
Emi Kurimoto
Takayuki Kawai
Minoru Maruyama
Hidetoshi Komatsu
Kensuke Sakuma
Yuji Shimizu
Masato Shimojo
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Citations (15)
Discovery of the First Potent and Orally Available Agonist of the Orphan G-Protein-Coupled Receptor 52
2014
Journal of Medicinal Chemistry
Masaki Setoh
Naoki Ishii
Mitsunori Kono
Yuhei Miyanohana
Eri Shiraishi
Toshiya Harasawa
Hiroyuki Ota
Tomoyuki Odani
Naoyuki Kanzaki
Kazunobu Aoyama
Teruki Hamada
Masakuni Kori
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Citations (27)
1