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Hiroki Takahagi
Hiroki Takahagi
Takeda Pharmaceutical Company
Biochemistry
Chemistry
Trifluoromethyl
Organic chemistry
Acyl-CoA
3
Papers
41
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A pyridone derivative activates SERCA2a by attenuating the inhibitory effect of phospholamban
2017
European Journal of Pharmacology
Manami Kaneko
Hisato Yamamoto
Hiroki Sakai
Yusuke Kamada
Toshiki Tanaka
Shuji Fujiwara
Syunsuke Yamamoto
Hiroki Takahagi
Hideyuki Igawa
Shizuo Kasai
Masakuni Noda
Makoto Inui
Tomoyuki Nishimoto
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Citations (8)
Discovery of a Novel Series of N-Phenylindoline-5-sulfonamide Derivatives as Potent, Selective, and Orally Bioavailable Acyl CoA:Monoacylglycerol Acyltransferase-2 Inhibitors
2015
Journal of Medicinal Chemistry
Kenjiro Sato
Hiroki Takahagi
Takeshi Yoshikawa
Shinji Morimoto
Takafumi Takai
Kousuke Hidaka
Masahiro Kamaura
Osamu Kubo
Ryutaro Adachi
Tsuyoshi Ishii
Toshiyuki Maki
Taisuke Mochida
Shiro Takekawa
Masanori Nakakariya
Nobuyuki Amano
Tomoyuki Kitazaki
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Citations (25)
Optimization of a novel series of N-phenylindoline-5-sulfonamide-based acyl CoA:monoacylglycerol acyltransferase-2 inhibitors: Mitigation of CYP3A4 time-dependent inhibition and phototoxic liabilities
2015
Bioorganic & Medicinal Chemistry
Kenjiro Sato
Hiroki Takahagi
Osamu Kubo
Kousuke Hidaka
Takeshi Yoshikawa
Masahiro Kamaura
Masanori Nakakariya
Nobuyuki Amano
Ryutaro Adachi
Toshiyuki Maki
Kazumi Take
Shiro Takekawa
Tomoyuki Kitazaki
Tsuyoshi Maekawa
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Citations (8)
1