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Giuseppe Marseglia
Giuseppe Marseglia
University of Parma
Chemistry
Stereochemistry
Fibroblast growth factor receptor
Cancer research
Fibroblast growth factor
4
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11
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Chemical modification of NSC12 leads to a specific FGF-trap with antitumor activity in multiple myeloma.
2021
European Journal of Medicinal Chemistry
Riccardo Castelli
Sara Taranto
Lucia Furiassi
Nicole Bozza
Giuseppe Marseglia
Francesca Ferlenghi
Silvia Rivara
Michele Retini
Annalida Bedini
Gilberto Spadoni
Sara Matarazzo
Roberto Ronca
Marco Presta
Marco Mor
Arianna Giacomini
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A sulfonyl fluoride derivative inhibits EGFRL858R/T790M/C797S by covalent modification of the catalytic lysine.
2021
European Journal of Medicinal Chemistry
Francesca Ferlenghi
Laura Scalvini
Federica Vacondio
Riccardo Castelli
Nicole Bozza
Giuseppe Marseglia
Silvia Rivara
Alessio Lodola
Silvia La Monica
Roberta Minari
Pier Giorgio Petronini
Roberta Alfieri
Marcello Tiseo
Marco Mor
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Deconstructing Noncovalent Kelch-like ECH-Associated Protein 1 (Keap1) Inhibitors into Fragments to Reconstruct New Potent Compounds.
2021
Journal of Medicinal Chemistry
Jakob S. Pallesen
Dilip Narayanan
Kim T. Tran
Sara Marie Øie Solbak
Giuseppe Marseglia
Louis M.E. Sørensen
Lars Jakobsen Høj
Federico Munafò
Rosa M. C. Carmona
Anthony D. Garcia
Haritha L. Desu
Roberta Brambilla
Tommy N. Johansen
Grzegorz M. Popowicz
Michael Sattler
Michael Gajhede
Anders Bach
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Fibroblast growth factor receptor inhibitors: patent review (2015–2019)
2019
Expert Opinion on Therapeutic Patents
Giuseppe Marseglia
Alessio Lodola
Marco Mor
Riccardo Castelli
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Citations (6)
1