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Hikari Araki
Hikari Araki
Cancer research
Immunology
Medicine
Covalent bond
Molecular biology
4
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5
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0
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TAS0728, A Covalent-binding, HER2-selective Kinase Inhibitor Shows Potent Antitumor Activity in Preclinical Models
2019
Molecular Cancer Therapeutics
Hiroki Irie
Kimihiro Ito
Yayoi Fujioka
Kei Oguchi
Akio Fujioka
Akihiro Hashimoto
Hirokazu Ohsawa
Kenji Tanaka
Kaoru Funabashi
Hikari Araki
Yuichi Kawai
Tadashi Shimamura
Renu Wadhwa
Shuichi Ohkubo
Kenichi Matsuo
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Abstract B179: TAS0728, a HER2-selective covalent inhibitor, demonstrates potent antitumor effect as a single agent and in combination with anti-HER2 antibodies in HER2-overexpressed tumor models
2018
Molecular Cancer Therapeutics
Hiroki Irie
Kei Oguchi
Kimihiro Ito
Yayoi Fujioka
Yuichi Kawai
Tadashi Shimamura
Hikari Araki
Akio Fujioka
Fumio Nakagawa
Rumi Kawabata
Hideki Nagase
Takeshi Sagara
Junji Uchida
Kenichi Matsuo
Teruhiro Utsugi
Yoshikazu Iwasawa
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TPC-107, a next generation, HER2 selective covalent inhibitor demonstrates potent inhibition for activated mutations of HER2 while sparing EGFR inhibition
2016
European Journal of Cancer
Kei Oguchi
Hiroki Irie
Kimihiro Ito
Yayoi Fujioka
Yuji Yamada
Tadashi Shimamura
Yuichi Kawai
Yoshihiro Shibata
Hikari Araki
Tomonori Haruma
Akio Fujioka
Takeshi Sagara
Kenichi Matsuo
Teruhiro Utsugi
Yoshikazu Iwasawa
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TPC-107, a next generation, HER2 selective covalent inhibitor demonstrates potent and sustained inhibition against the HER2–HER3 signaling while sparing EGFR activity, leading to a large therapeutic window
2016
European Journal of Cancer
Hiroki Irie
Kimihiro Ito
Y. Kataoka
Yayoi Fujioka
Kei Oguchi
Tadashi Shimamura
Yuichi Kawai
Takeshi Sagara
Yoshihiro Shibata
Hikari Araki
Tomonori Haruma
Akihiro Hashimoto
Kenichi Matsuo
Teruhiro Utsugi
Yoshikazu Iwasawa
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