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Mihaela-Liliana Ţînţaş
Mihaela-Liliana Ţînţaş
Centre national de la recherche scientifique
Chemistry
Prodrug
Organic chemistry
Serine
Docking (molecular)
3
Papers
25
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Rational design of carbamate-based dual binding site and central AChE inhibitors by a “biooxidisable” prodrug approach: Synthesis, in vitro evaluation and docking studies
2018
European Journal of Medicinal Chemistry
Mihaela-Liliana Ţînţaş
Vincent Gembus
Florent Alix
Anaïs Barré
Gaël Coadou
Lina Truong
Muriel Sebban
Cyril Papamicaël
Hassan Oulyadi
Vincent Levacher
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Citations (3)
Access to Highly Enantioenriched Donepezil-like 1,4-Dihydropyridines as Promising Anti-Alzheimer Prodrug Candidates via Enantioselective Tsuji Allylation and Organocatalytic Aza-Ene-Type Domino Reactions
2018
Journal of Organic Chemistry
Mihaela-Liliana Ţînţaş
Rabah Azzouz
Ludovic Peauger
Vincent Gembus
Emilie Petit
Laëtitia Bailly
Cyril Papamicaël
Vincent Levacher
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Citations (5)
Palladium-Catalyzed Carbonylation of (Hetero)Aryl, Alkenyl and Allyl Halides by Means of N-Hydroxysuccinimidyl Formate as CO Surrogate
2015
Journal of Organic Chemistry
Anaïs Barré
Mihaela-Liliana Ţînţaş
Florent Alix
Vincent Gembus
Cyril Papamicaël
Vincent Levacher
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Citations (17)
1