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Lina Truong
Lina Truong
Centre national de la recherche scientifique
Prodrug
Carbamate
Chemistry
Safety pharmacology
Acetylcholinesterase inhibitor
2
Papers
6
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0
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Rational design of carbamate-based dual binding site and central AChE inhibitors by a “biooxidisable” prodrug approach: Synthesis, in vitro evaluation and docking studies
2018
European Journal of Medicinal Chemistry
Mihaela-Liliana Ţînţaş
Vincent Gembus
Florent Alix
Anaïs Barré
Gaël Coadou
Lina Truong
Muriel Sebban
Cyril Papamicaël
Hassan Oulyadi
Vincent Levacher
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Citations (3)
Dihydroquinoline Carbamate DQS1-02 as a Prodrug of a Potent Acetylcholinesterase Inhibitor for Alzheimer’s Disease Therapy: Multigram-Scale Synthesis, Mechanism Investigations, in Vitro Safety Pharmacology, and Preliminary in Vivo Toxicology Profile
2018
Florent Alix
Vincent Gembus
Laurent Coquet
Marie Hubert-Roux
Philippe Chan
Lina Truong
Muriel Sebban
Gaël Coadou
Hassan Oulyadi
Cyril Papamicaël
Vincent Levacher
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Citations (3)
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