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Toshiki Murata
Toshiki Murata
Takeda Pharmaceutical Company
Stereochemistry
Chemistry
Indoline
hERG
Agonist
4
Papers
34
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2024
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Discovery of a Novel Series of Indolinylpyrimidine-based GPR119 Agonists: Elimination of Ether-a-go-go-related Gene Liability Using a Hydrogen Bond acceptor-Focused Approach
2021
Bioorganic & Medicinal Chemistry
Masahiro Kamaura
Osamu Kubo
Hiromichi Sugimoto
Naoyoshi Noguchi
Hirohisa Miyashita
Shin-Ichi Abe
Kae Matsuda
Yoshiyuki Tsujihata
Tomoyuki Odani
Shinji Iwasaki
Toshiki Murata
Kenjiro Sato
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Citations (1)
Discovery of a novel series of GPR119 agonists: Design, synthesis, and biological evaluation of N-(Piperidin-4-yl)-N-(trifluoromethyl)pyrimidin-4-amine derivatives.
2021
Bioorganic & Medicinal Chemistry
Osamu Kubo
Kazuaki Takami
Masahiro Kamaura
Koji Watanabe
Hirohisa Miyashita
Shin-Ichi Abe
Kae Matsuda
Yoshiyuki Tsujihata
Tomoyuki Odani
Shinji Iwasaki
Tomoyuki Kitazaki
Toshiki Murata
Kenjiro Sato
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Discovery of a novel series of indoline carbamate and indolinylpyrimidine derivatives as potent GPR119 agonists.
2014
Bioorganic & Medicinal Chemistry
Kenjiro Sato
Hiromichi Sugimoto
Kentaro Rikimaru
Hiroshi Imoto
Masahiro Kamaura
Nobuyuki Negoro
Yoshiyuki Tsujihata
Hirohisa Miyashita
Tomoyuki Odani
Toshiki Murata
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Citations (20)
Synthesis, Structure–Activity Relationship, and Pharmacological Studies of Novel Melanin-Concentrating Hormone Receptor 1 Antagonists 3-Aminomethylquinolines: Reducing Human Ether-a-go-go-Related Gene (hERG) Associated Liabilities
2012
Journal of Medicinal Chemistry
Shizuo Kasai
Makoto Kamata
Shinichi Masada
Jun Kunitomo
Masahiro Kamaura
Tomohiro Okawa
Kazuaki Takami
Hitomi Ogino
Yoshihide Nakano
Shuntarou Ashina
Kaoru Watanabe
Tomoko Kaisho
Yumi N. Imai
Sunghi Ryu
Masaharu Nakayama
Yasutaka Nagisa
Shiro Takekawa
Koki Kato
Toshiki Murata
Nobuhiro Suzuki
Yuji Ishihara
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Citations (13)
1