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Shin-Ichi Abe
Shin-Ichi Abe
Takeda Pharmaceutical Company
Chemistry
Agonist
Receptor
hERG
Stereochemistry
3
Papers
10
Citations
0
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2024
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Discovery of a Novel Series of Indolinylpyrimidine-based GPR119 Agonists: Elimination of Ether-a-go-go-related Gene Liability Using a Hydrogen Bond acceptor-Focused Approach
2021
Bioorganic & Medicinal Chemistry
Masahiro Kamaura
Osamu Kubo
Hiromichi Sugimoto
Naoyoshi Noguchi
Hirohisa Miyashita
Shin-Ichi Abe
Kae Matsuda
Yoshiyuki Tsujihata
Tomoyuki Odani
Shinji Iwasaki
Toshiki Murata
Kenjiro Sato
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Citations (1)
Discovery of a novel series of GPR119 agonists: Design, synthesis, and biological evaluation of N-(Piperidin-4-yl)-N-(trifluoromethyl)pyrimidin-4-amine derivatives.
2021
Bioorganic & Medicinal Chemistry
Osamu Kubo
Kazuaki Takami
Masahiro Kamaura
Koji Watanabe
Hirohisa Miyashita
Shin-Ichi Abe
Kae Matsuda
Yoshiyuki Tsujihata
Tomoyuki Odani
Shinji Iwasaki
Tomoyuki Kitazaki
Toshiki Murata
Kenjiro Sato
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GPR40 full agonism exerts feeding suppression and weight loss through afferent vagal nerve
2019
PLOS ONE
Hikaru Ueno
Ryo Ito
Shin-Ichi Abe
Hitomi Ogino
Minoru Maruyama
Hirohisa Miyashita
Yasufumi Miyamoto
Yusuke Moritoh
Yoshiyuki Tsujihata
Koji Takeuchi
Nobuhiro Nishigaki
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Citations (9)
1