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Brian T. Masick
Brian T. Masick
Genomics Institute of the Novartis Research Foundation
Chemistry
Biochemistry
Stereochemistry
Organic chemistry
Enzyme
4
Papers
118
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Discovery, Optimization, and Biological Evaluation of 5-(2-(Trifluoromethyl)phenyl)indazoles as a Novel Class of Transient Receptor Potential A1 (TRPA1) Antagonists
2014
Journal of Medicinal Chemistry
Lisa Rooney
Agnes Vidal
Anne-Marie D’Souza
Nicholas James Devereux
Brian T. Masick
Valerie Boissel
Ryan West
Victoria Head
Rowan Stringer
Jianmin Lao
Matt Petrus
Ardem Patapoutian
Mark Nash
Natalie Stoakley
Moh Panesar
J. Martin Verkuyl
Andrew Schumacher
H. Michael Petrassi
David C. Tully
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Citations (32)
Substrate optimization for monitoring cathepsin C activity in live cells
2009
Bioorganic & Medicinal Chemistry
Jun Li
H. Michael Petrassi
Christine Tumanut
Brian T. Masick
Christopher Trussell
Jennifer L. Harris
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Citations (18)
Synthesis and SAR of arylaminoethyl amides as noncovalent inhibitors of cathepsin S: P3 cyclic ethers.
2006
Bioorganic & Medicinal Chemistry Letters
David C. Tully
Hong Liu
Arnab K. Chatterjee
Phil B. Alper
Robert Epple
Jennifer A. Williams
Michael J. Roberts
David H. Woodmansee
Brian T. Masick
Christine Tumanut
Jun Li
Glen Spraggon
Michael Hornsby
Jonathan Chang
Tove Tuntland
Thomas Hollenbeck
Perry Gordon
Jennifer L. Harris
Donald S. Karanewsky
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Citations (28)
A strategy to profile prime and non-prime proteolytic substrate specificity
2005
Bioorganic & Medicinal Chemistry Letters
H. Michael Petrassi
Jennifer A. Williams
Jun Li
Christine Tumanut
Jared Ek
Takashi Nakai
Brian T. Masick
Bradley J. Backes
Jennifer L. Harris
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Citations (40)
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