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Valerie Boissel
Valerie Boissel
Novartis
Chemistry
Trifluoromethyl
Hit to lead
Antagonist
Indazole
2
Papers
32
Citations
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Discovery, Optimization, and Biological Evaluation of 5-(2-(Trifluoromethyl)phenyl)indazoles as a Novel Class of Transient Receptor Potential A1 (TRPA1) Antagonists
2014
Journal of Medicinal Chemistry
Lisa Rooney
Agnes Vidal
Anne-Marie D’Souza
Nicholas James Devereux
Brian T. Masick
Valerie Boissel
Ryan West
Victoria Head
Rowan Stringer
Jianmin Lao
Matt Petrus
Ardem Patapoutian
Mark Nash
Natalie Stoakley
Moh Panesar
J. Martin Verkuyl
Andrew Schumacher
H. Michael Petrassi
David C. Tully
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Citations (32)
Synthesis of drug-like molecules for respiratory diseases: utilizing microwave chemistry
2014
Valerie Boissel
Rebecca Butler
Paul J Oakley
Neil J Press
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