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Guanghui Deng
Guanghui Deng
GlaxoSmithKline
Chemistry
Biochemistry
Oral administration
Agonist
In vivo
4
Papers
52
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Novel complex crystal structure of prolyl hydroxylase domain-containing protein 2 (PHD2): 2,8-Diazaspiro[4.5]decan-1-ones as potent, orally bioavailable PHD2 inhibitors
2013
Bioorganic & Medicinal Chemistry
Guanghui Deng
Baowei Zhao
Yingli Ma
Qiongfeng Xu
Hailong Wang
Liuqing Yang
Qing Zhang
Taylor B. Guo
Wei Zhang
Yang Jiao
Xin Cai
Jinqiang Zhang
Houfu Liu
Xiaoming Guan
Hongtao Lu
Jia-Ning Xiang
John D. Elliott
Xichen Lin
Feng Ren
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Citations (14)
Identification of benzoxazole analogs as novel, S1P3 sparing S1P1 agonists
2012
Bioorganic & Medicinal Chemistry Letters
Guanghui Deng
Qinghua Meng
Qian Liu
Xuesong Xu
Qiongfeng Xu
Feng Ren
Taylor B. Guo
Hongtao Lu
Jia-Ning Xiang
John D. Elliott
Xichen Lin
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Citations (6)
Discovery of Novel 1,2,4-Thiadiazole Derivatives as Potent, Orally Active Agonists of Sphingosine 1-Phosphate Receptor Subtype 1 (S1P1)
2012
Journal of Medicinal Chemistry
Feng Ren
Guanghui Deng
Hailong Wang
Linbo Luan
Qinghua Meng
Qiongfeng Xu
Heng Xu
Xuesong Xu
Haibo Zhang
Baowei Zhao
Chengyong Li
Taylor B. Guo
Jiansong Yang
Wei Zhang
Yonggang Zhao
Qiantao Jia
Hongtao Lu
Jia-Ning Xiang
John D. Elliott
Xichen Lin
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Citations (22)
Indole-propionic acid derivatives as potent, S1P3-sparing and EAE efficacious sphingosine-1-phosphate 1 (S1P1) receptor agonists.
2012
Bioorganic & Medicinal Chemistry Letters
Qinghua Meng
Baowei Zhao
Qiongfeng Xu
Xuesong Xu
Guanghui Deng
Chengyong Li
Linbo Luan
Feng Ren
Hailong Wang
Heng Xu
Yan Xu
Haibo Zhang
Jia-Ning Xiang
John D. Elliott
Taylor B. Guo
Yonggang Zhao
Wei Zhang
Hongtao Lu
Xichen Lin
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Citations (10)
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