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Toshifumi Tojo
Toshifumi Tojo
Kyoto Prefectural University of Medicine
Biochemistry
Chemistry
Demethylase
Histone
Stereochemistry
3
Papers
68
Citations
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Identification of Diketopiperazine-Containing 2-Anilinobenzamides as Potent Sirtuin 2 (SIRT2)-Selective Inhibitors Targeting the “Selectivity Pocket”, Substrate-Binding Site, and NAD+-Binding Site
2019
Journal of Medicinal Chemistry
Paolo Mellini
Yukihiro Itoh
Elghareeb E. Elboray
Hiroki Tsumoto
Ying Li
Miki Suzuki
Yukari Takahashi
Toshifumi Tojo
Takashi Kurohara
Yuka Miyake
Yuri Miura
Yuki Kitao
Masayuki Kotoku
Tetsuya Iida
Takayoshi Suzuki
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Citations (10)
Identification of SNAIL1 Peptide-Based Irreversible Lysine-Specific Demethylase 1-Selective Inactivators
2016
Journal of Medicinal Chemistry
Yukihiro Itoh
Keisuke Aihara
Paolo Mellini
Toshifumi Tojo
Yosuke Ota
Hiroki Tsumoto
Viswas Raja Solomon
Peng Zhan
Miki Suzuki
Daisuke Ogasawara
Akira Shigenaga
Tsubasa Inokuma
Hidehiko Nakagawa
Naoki Miyata
Tamio Mizukami
Akira Otaka
Takayoshi Suzuki
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Citations (20)
Identification of Jumonji AT-Rich Interactive Domain 1A Inhibitors and Their Effect on Cancer Cells
2015
ACS Medicinal Chemistry Letters
Yukihiro Itoh
Hideyuki Sawada
Miki Suzuki
Toshifumi Tojo
Ryuzo Sasaki
Makoto Hasegawa
Tamio Mizukami
Takayoshi Suzuki
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Citations (38)
1