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Takashi Sasaki
Takashi Sasaki
Mitsubishi Tanabe Pharma
Phosphodiesterase
PDE10A
Internal medicine
Endocrinology
Pyrimidine
4
Papers
291
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Discovery of a pyrazolo[1,5-a]pyrimidine derivative (MT-3014) as a highly selective PDE10A inhibitor via core structure transformation from the stilbene moiety
2019
Bioorganic & Medicinal Chemistry
Yuuki Koizumi
Yoshihito Tanaka
Takehiko Matsumura
Yoichi Kadoh
Haruko Miyoshi
Mitsuya Hongu
Kei Takedomi
Jun Kotera
Takashi Sasaki
Hiroyuki Taniguchi
Yumi Watanabe
Misae Takakuwa
Koki Kojima
Nobuyuki Baba
Itsuko Nakamura
Eiji Kawanishi
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Citations (6)
Discovery of 2-[(E)-2-(7-fluoro-3-methylquinoxalin-2-yl)vinyl]-6-pyrrolidin- 1-yl-N-(tetrahydro-2H-pyran-4-yl)pyrimidin-4-amine hydrochloride as a highly selective PDE10A inhibitor
2018
Chemical & Pharmaceutical Bulletin
Yoichi Kadoh
Haruko Miyoshi
Takehiko Matsumura
Yoshihito Tanaka
Mitsuya Hongu
Mayumi Kimura
Kei Takedomi
Kenji Omori
Jun Kotera
Takashi Sasaki
Tamaki Kobayashi
Hiroyuki Taniguchi
Yumi Watanabe
Koki Kojima
Toshiaki Sakamoto
Toshiyuki Himiyama
Eiji Kawanishi
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Citations (6)
Phosphodiesterase 9A controls nitric-oxide-independent cGMP and hypertrophic heart disease.
2015
Nature
Dong I. Lee
Guangshuo Zhu
Takashi Sasaki
Gun Sik Cho
Nazha Hamdani
Ronald J. Holewinski
Su-Hyun Jo
Thomas Danner
Manling Zhang
Peter P. Rainer
Djahida Bedja
Jonathan A. Kirk
Mark J. Ranek
Wolfgang R. Dostmann
Chulan Kwon
Kenneth B. Margulies
Jennifer E. Van Eyk
Walter Paulus
Eiki Takimoto
David A. Kass
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Citations (222)
Avanafil, a Potent and Highly Selective Phosphodiesterase-5 Inhibitor for Erectile Dysfunction
2012
The Journal of Urology
Jun Kotera
Hideki Mochida
Hirotaka Inoue
Tsunehisa Noto
Kotomi Fujishige
Takashi Sasaki
Tamaki Kobayashi
Koki Kojima
Shiyin Yee
Yasuhiro Yamada
Kohei Kikkawa
Kenji Omori
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Citations (57)
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