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Haruko Miyoshi
Haruko Miyoshi
Mitsubishi Tanabe Pharma
Pyrimidine
Organic chemistry
Quinoxaline
Chemistry
Stereochemistry
2
Papers
12
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2024
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Discovery of a pyrazolo[1,5-a]pyrimidine derivative (MT-3014) as a highly selective PDE10A inhibitor via core structure transformation from the stilbene moiety
2019
Bioorganic & Medicinal Chemistry
Yuuki Koizumi
Yoshihito Tanaka
Takehiko Matsumura
Yoichi Kadoh
Haruko Miyoshi
Mitsuya Hongu
Kei Takedomi
Jun Kotera
Takashi Sasaki
Hiroyuki Taniguchi
Yumi Watanabe
Misae Takakuwa
Koki Kojima
Nobuyuki Baba
Itsuko Nakamura
Eiji Kawanishi
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Discovery of 2-[(E)-2-(7-fluoro-3-methylquinoxalin-2-yl)vinyl]-6-pyrrolidin- 1-yl-N-(tetrahydro-2H-pyran-4-yl)pyrimidin-4-amine hydrochloride as a highly selective PDE10A inhibitor
2018
Chemical & Pharmaceutical Bulletin
Yoichi Kadoh
Haruko Miyoshi
Takehiko Matsumura
Yoshihito Tanaka
Mitsuya Hongu
Mayumi Kimura
Kei Takedomi
Kenji Omori
Jun Kotera
Takashi Sasaki
Tamaki Kobayashi
Hiroyuki Taniguchi
Yumi Watanabe
Koki Kojima
Toshiaki Sakamoto
Toshiyuki Himiyama
Eiji Kawanishi
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Citations (6)
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