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Yan Chen
Yan Chen
GlaxoSmithKline
Chemistry
Pharmacology
Pharmacokinetics
Bioavailability
Disposition
4
Papers
20
Citations
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5-Substituted-N-pyridazinylbenzamides as potent and selective LRRK2 inhibitors: Improved brain unbound fraction enables efficacy
2019
Bioorganic & Medicinal Chemistry Letters
Xiao Ding
Luigi Piero Stasi
Xuedong Dai
Kai Long
Cheng Peng
Baowei Zhao
Hailong Wang
Changhui Sun
Huan Hu
Zehong Wan
Karamjit Singh Jandu
Oliver James Philps
Yan Chen
Lizhen Wang
Qian Liu
Colin Edge
Yi Li
Kelly Dong
Xiaoming Guan
F. David Tattersall
Alastair D. Reith
Feng Ren
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Citations (3)
Rapid Bioavailability and Disposition protocol: A novel higher throughput approach to assess pharmacokinetics and steady-state brain distribution with reduced animal usage
2018
European Journal of Pharmaceutical Sciences
Tingting Fu
Ruina Gao
Paul Scott-Stevens
Yan Chen
Chalmers Zhang
Jianfei Wang
Scott Summerfield
Houfu Liu
Jasminder Sahi
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Citations (1)
Drug Distribution into Peripheral Nerve
2018
Journal of Pharmacology and Experimental Therapeutics
Houfu Liu
Yan Chen
Liang Huang
Xueying Sun
Tingting Fu
Shengqian Wu
Xiaoyan Zhu
Wei Zhen
Jihong Liu
Gang Lu
Wei Cai
Ting Yang
Wandong Zhang
Xiaohong Yu
Zehong Wan
Jianfei Wang
Scott Summerfield
Kelly Dong
Georg C. Terstappen
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Citations (16)
Rapid bioavailability and disposition protocol: A novel higher throughput approach to assess pharmacokinetics and steady-state tissue disstribution using fewer animals
2017
Drug Metabolism and Pharmacokinetics
Tingting Fu
Ruina Gao
Paul Scott-Stevens
Yan Chen
Chalmers Zhang
Jianfei Wang
Scott Summerfield
Valeriu Damian
Jasminder Sahi
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