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Alastair D. Reith
Alastair D. Reith
The Hertz Corporation
Biochemistry
LRRK2
Chemistry
Kinase
Kinome
3
Papers
18
Citations
0
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2024
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5-Substituted-N-pyridazinylbenzamides as potent and selective LRRK2 inhibitors: Improved brain unbound fraction enables efficacy
2019
Bioorganic & Medicinal Chemistry Letters
Xiao Ding
Luigi Piero Stasi
Xuedong Dai
Kai Long
Cheng Peng
Baowei Zhao
Hailong Wang
Changhui Sun
Huan Hu
Zehong Wan
Karamjit Singh Jandu
Oliver James Philps
Yan Chen
Lizhen Wang
Qian Liu
Colin Edge
Yi Li
Kelly Dong
Xiaoming Guan
F. David Tattersall
Alastair D. Reith
Feng Ren
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Citations (3)
Discovery of 4-ethoxy-7H-pyrrolo[2,3-d]pyrimidin-2-amines as potent, selective and orally bioavailable LRRK2 inhibitors
2018
Bioorganic & Medicinal Chemistry Letters
Xiao Ding
Luigi Piero Stasi
Ming-Hsun Ho
Baowei Zhao
Hailong Wang
Kai Long
Qiongfeng Xu
Yingxia Sang
Changhui Sun
Huan Hu
Haihua Yu
Zehong Wan
Lizhen Wang
Colin Edge
Qian Liu
Yi Li
Kelly Dong
Xiaoming Guan
F. David Tattersall
Alastair D. Reith
Feng Ren
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Citations (6)
Discovery of 5-substituent-N-arylbenzamide derivatives as potent, selective and orally bioavailable LRRK2 inhibitors
2017
Bioorganic & Medicinal Chemistry Letters
Xiao Ding
Xuedong Dai
Kai Long
Cheng Peng
Daniele Andreotti
Paul Bamborough
Andrew John Eatherton
Colin Edge
Karamjit Singh Jandu
Paula Louise Nichols
Oliver James Philps
Luigi Piero Stasi
Zehong Wan
Jia-Ning Xiang
Kelly Dong
Pamela Dossang
Ming-Hsun Ho
Yi Li
Lucy M. Mensah
Xiaoming Guan
Alastair D. Reith
Feng Ren
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Citations (9)
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