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Imelda Lam
Imelda Lam
Cereblon
Homeostasis
Medicine
Cell biology
Cancer research
4
Papers
2
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0
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Abstract 1963: Targeting hematological malignancies with two functionally and mechanistically distinct classes of cereblon mediated protein homeostatic modulators
2020
Aparajita Hoskote Chourasia
Leah Fung
Angela Pasis
Brooke McElwee
Angela Schoolmeesters
Normand Richard
Imelda Lam
Eduardo Torres
Paul Erdman
Sullivan Robert
David Hecht
Kyle W. H. Chan
Frank Mercurio
David I. Stirling
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Citations (1)
The novel protein homeostatic modulator BTX306 is active in myeloma and overcomes bortezomib and lenalidomide resistance.
2020
Journal of Molecular Medicine
Jianxuan Zou
Richard J. Jones
Hua Wang
Isere Kuiatse
Fazal Shirazi
Elisabet E. Manasanch
Hans C. Lee
Robert W. Sullivan
Leah Fung
Normand Richard
Paul Erdman
Eduardo Torres
David Hecht
Imelda Lam
Brooke McElwee
Aparajita Hoskote Chourasia
Kyle W. H. Chan
Frank Mercurio
David I. Stirling
Robert Z. Orlowski
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Bioavailable Dual-Protein Degraders of CK1α and Transcriptional Kinase CDK9 As Potential Therapeutics for Hematological Malignancies
2019
Blood
Leah Fung
Aparajita Hoskote Chourasia
Eduardo Torres
Imelda Lam
Paul Erdman
David Hecht
Robert W. Sullivan
Brooke McElwee
Normand Richard
Avanthika Venkatachalam
Irit Snir-Alkalay
Kyle W. H. Chan
Frank Mercurio
Yinon Ben Neriah
David I. Stirling
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Targeting AML: The Development of Two Functionally and Mechanistically Distinct Classes of Cereblon-Mediated Protein Homeostatic Modulators
2019
Blood
Aparajita Hoskote Chourasia
Leah Fung
Brooke McElwee
Normand Richard
Imelda Lam
Eduardo Torres
Paul Erdman
Robert W. Sullivan
David Hecht
Kyle W. H. Chan
Frank Mercurio
David I. Stirling
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